Optimization of Hydroxyethylamine Transition State Isosteres as Aspartic Protease Inhibitors by Exploiting Conformational Preferences

  1. Bueno, A.B.
  2. Agejas, J.
  3. Broughton, H.
  4. Dally, R.
  5. Durham, T.B.
  6. Espinosa, J.F.
  7. González, R.
  8. Hahn, P.J.
  9. Marcos, A.
  10. Rodríguez, R.
  11. Sanz, G.
  12. Soriano, J.F.
  13. Timm, D.
  14. Vidal, P.
  15. Yang, H.-C.
  16. McCarthy, J.R.
Aldizkaria:
Journal of Medicinal Chemistry

ISSN: 1520-4804 0022-2623

Argitalpen urtea: 2017

Alea: 60

Zenbakia: 23

Orrialdeak: 9807-9820

Mota: Artikulua

DOI: 10.1021/ACS.JMEDCHEM.7B01304 GOOGLE SCHOLAR