Discovery of EST73502, a Dual μ-Opioid Receptor Agonist and σ1Receptor Antagonist Clinical Candidate for the Treatment of Pain

  1. García, M.
  2. Virgili, M.
  3. Alonso, M.
  4. Alegret, C.
  5. Farran, J.
  6. Fernández, B.
  7. Bordas, M.
  8. Pascual, R.
  9. Burgueño, J.
  10. Vidal-Torres, A.
  11. Fernández De Henestrosa, A.R.
  12. Ayet, E.
  13. Merlos, M.
  14. Vela, J.M.
  15. Plata-Salamán, C.R.
  16. Almansa, C.
Journal:
Journal of Medicinal Chemistry

ISSN: 1520-4804 0022-2623

Year of publication: 2020

Volume: 63

Issue: 24

Pages: 15508-15526

Type: Article

DOI: 10.1021/ACS.JMEDCHEM.0C01127 GOOGLE SCHOLAR