Publikationen in Zusammenarbeit mit Forschern von Eli Lilly and Company (4)

2017

  1. Optimization of Hydroxyethylamine Transition State Isosteres as Aspartic Protease Inhibitors by Exploiting Conformational Preferences

    Journal of Medicinal Chemistry, Vol. 60, Núm. 23, pp. 9807-9820

2005

  1. 2-Alkoxydihydrocinnamates as PPAR agonists. Activity modulation by the incorporation of phenoxy substituents

    Bioorganic and Medicinal Chemistry Letters, Vol. 15, Núm. 1, pp. 51-55

2004

  1. (2S,1′S,2′R,3′R)-2-(2′-Carboxy-3′ -hydroxymethylcyclopropyl) Glycine Is a Highly Potent Group 2 and 3 Metabotropic Glutamate Receptor Agonist with Oral Activity

    Journal of Medicinal Chemistry, Vol. 47, Núm. 2, pp. 456-466

1995

  1. Conformationally constrained ACPD analogues. Synthesis and resolution of 3-aminobicyclo[3,3,0]octane-1,3-dicarboxylic acids

    Tetrahedron, Vol. 51, Núm. 11, pp. 3271-3278